Izenzo zeMithi yeMithi yokuVimbela i-Orexin kwiBrain
Isichengululo seziyobisi esithengiswayo phantsi kwegama lophawu lweBelsomra-liyimpilisi yokulala ekhethiweyo esetyenziswayo ukuphatha ingxaki ehla okanye ukulala ubuthongo obonakalisa ukulala . Funda malunga nendlela esebenza ngayo kunye nezinye iziphumo ezibi kunye neengozi ezinxulumene nokusetyenziswa kweBelsomra.
Ukusetyenziswa kweBelsomra
I-Belsomra yonyango lonyango elisebenza kwingqondo ukunciphisa ukuvuka nokuphucula ubuthongo.
Kubangela ukulala nokusebenza ngokufanelekileyo ukuqala nokugcina ubuthongo. Isetyenziswe ngokuyinhloko ukunyanga ukulala. Kubonakala kunenzuzo ethobekileyo kubantu abaninzi abanomdla obonisa ukuba abantu abalalayo balala bemizuzu engama-6 ngokukhawuleza kwaye balala nje imizuzu eyi-16 kuphela, xa kuthelekiswa ne-placebo.
I-Belsomra isebenze njani ukuphathwa ngongqungquthela?
I-Belsomra iyingqayizivele phakathi kokulala kweepilisi ngendlela isebenza ngayo. Ukuvunyelwa yi-US Food Administration and Drug Administration ngo-2014, ngowokuqala kwiklasi yamayeza asebenza njenge- orexin . I-Orexin i-neurotransmitter, okanye umthunywa weekhemikhali, ngaphakathi kwengqondo ekhuthaza ukuvuka. Xa ivinjiwe, njengokuba kwenzeka nakubandezeli, ubuthongo bungabangela.
I-Belsomra ikhethe kakhulu i-receptors yamagunya ebizwa nge-OX1R ne-OX2R ngaphakathi kwengqondo. Ngokuzibandakanya nala ma-receptors, unako ukuvimba izinto ezikhuthazayo ezibizwa ngokuthi yi-orexin A kunye ne-orexin B, eyokukhazamisa ukukwazi ukuhlala uphapheme.
Iimpawu ze-narcolepsy zenzeka ngenxa yokulahlekelwa ngonaphakade kwezi seli ze-orexin.
Ngubani ongayisebenzisi iBelsomra?
Kukho abantu abathile abamele bangasebenzisi iBelsomra okanye ngubani omele awusebenzise ngokuqaphela. Akufanele isetyenziswe ukuba unesiqhwenga . Kumele kuthathwe zingama-30 imizuzu yokulala kwaye akufanele isetyenziswe ukuba awukwazi ukunikela ngaphezu kweeyure ezingama-7 ukuze ulale.
Ukulumkisa okucetyiswayo xa unembali yokudakumba, ukugula kwengqondo, okanye iingcinga zokuzibulala. Akufanele isetyenziswe ngokudibanisa notywala okanye ezinye iziyobisi ezinqanda inkqubo yesantya okanye inkqubo yokuphefumula. Ukuba unembali yokusetyenziswa kakubi kweziyobisi okanye umlutha, akufanele usebenzise.
Abo baneengxaki zomphunga okanye zesibindi kufuneka baqaphele xa besisebenzisa. Abantu abangenayo kunye nabasetyhini banokufuna amayeza amancinci ukukhusela imiphumo emibi. Ngenxa yokungabikho kolwazi malunga nokulimala, akukhuthazwa ukuba kusetyenziswe ngabasetyhini abakhulelweyo okanye abancancisayo.
Ziziphi iimpawu eziqhelekileyo okanye ezibi kakhulu zeBelsomra?
Kukho imiphumo emininzi yemiphumo yonyango. Umphumo oqhelekileyo ochaphazelekayo ngeBelsomra ubuthongo. Nangona umntu mhlawumbi akanakuze abe nemiphumo emibi kakhulu echaphazelekayo kunye neziyobisi-kwaye akunakwenzeka ukuba ikhona - enye into eyenzeka ngeBelsomra ifaka:
- Ukulala, ukunyaniseka, okanye "inkunkuma"
- Ukuphaphazeka nokulungelelanisa, kubandakanywa umngcipheko wokuqhuba ukulala
- Ukucinga okungavamile kunye nokuguquka kokuziphatha (ukuphuma okanye ukuziphatha kakubi, ukudideka, ukuphazamiseka, ukulahlekelwa kwememori, ukuxhalabisa, kunye neengcinga )
- Ukuxinezeleka nokuxhalabisa
- Ukuziphatha okuxinene nokulala (ukuqhuba, ukutya, ukulala ngesondo, njl.).
- Ukulala ukukhubazeka (ukungakwazi ukuhamba ngexesha lokuguquka kokulala)
- Ubuthakathaka bomlenze wesikhashana (ofana ne- cataplexy ngaphandle kwe-trigger)
- Ukuphefumula okuxhamlekileyo
Yiyiphi Inqununu Yokukhusela Imfuneko Yokuthathwa NgeBelsomra?
Ngenxa yengozi engaziwayo, i-Belsomra kufuneka igwenywe ekukhuleleni nasekunceliseni. Abanye abantu, njengoko kuchazwe ngentla, kufuneka basebenzise amayeza ngokulumkisa okanye kungekhona. Akukho nongweni efunekayo yokusetyenziswa kweBelsomra.
Ukuba ufumana ubunzima, kufuneka ube kunye nobudlelwane obusondeleyo nomboneleli wezempilo oyintloko.
> Imithombo:
> "IBelsomra Information Prescription Full." Merck & Co., Inc. 2014.
> "IBelsomra yeWebhusayithi ye-Offline." Merck & Co., Inc. 2014.
> "I-FDA iyavuma uhlobo olutsha lwesilonda sokulala, iBelsomra." Ulawulo lwe-US nokuLawulwa kweeDrug . Agasti 13, 2014.