I-Picamilon isongezelelo sokutya esenziwe ngokuhlanganiswa kwe-niacin (eyaziwa ngokuba yi-vitamin B3) kunye ne- gamma-aminobutyric acid (GABA) . Ngamanye amaxesha ekubhekiswa kuthiwa yi-nicotinoyl-GABA, i-picamilon ithengiswa njengesigqirha semithi eRussia.
I-Niacin iyaziwa ngokukhuthaza ukwandiswa kwemithambo yegazi, ngelixa i-gamma-aminobutyric acid idlala indima ebalulekileyo ekulawuleni umsebenzi wenkqubo yesondlo.
I-amino acid itholakala ngokwemvelo emzimbeni wakho, i-GABA isebenza njenge-neurotransmitter (uhlobo lweekhemikhali olujongene nokuthwala ulwazi ukusuka kwelinye iseli ukuya kwelinye). Uphando lubonisa ukuba abantu abaneengxaki ezithile zempilo yengqondo (ezifana nokudakumba okukhulu kunye nokuxhalabisa) banakho amathuba okuba namazinga aphantsi e-GABA.
Ukusetyenziswa
I-Picamilon idla ngokubizwa ngokuthi "izidakamizwa ezikhethileyo," iklasi leziyobisi ezisetyenziselwa kwenye iyeza ukuze kuphuculwe ukusebenza kwengqondo. Ukongeza, i-picamilon kuthiwa uncede ukuphatha ezi zilandelayo:
- Ukuxhalabisa (kuquka ukuxhalaba kwabantu)
- Ukuxinezeleka
- Igazi elonyukayo
- Migraine
Ezinye iziphakamisi zonyango ezizezinye zithi i-picamilon inokukunceda ekuphuculeni imemori, ukukhuthaza isimo sengqondo, nokukhusela isifo se-Alzheimer.
Izinzuzo
Kuze kube ngoku, ezimbalwa izifundo zenzululwazi ziye zavavanya iziphumo zempilo ze-picamilon. Nangona kunjalo, uphando oluthile lubonisa ukuba i-picamilon inokunikela ngezibonelelo ezithile.
Ngokomzekelo, uphando olusekelwe kwikarashi olukhishwe yi-Kiev Institute of Biochemistry ngo-1998 lucacise ukuba i-picamilon ibonisa isithembiso sokonyango kunye nokuthintela ukukhubazeka kwesifo sikashukela (imeko ephawulwe ngumonakalo wamanxeba obangelwa kukuphakama kwesifo sikashukela- ehambisana nomgangatho wezinga legazi).
Nangona kunjalo, ngoku kukho ukungabikho kweemvavanyo zonyango kwiipilamilon iziphumo ezinxamnye ne-neuropathy ye-diabetes.
Ukongezelela, uphando olwenziwa ngo-2010 olupapashwe kwiphepha laseRashiya I- Experimental kunye ne-Clinical Pharmacology yafumanisa ukuba i-picamilon inokukunceda ukukhusela kwi-hypokinesia. Kwiimvavanyo kwierati, abalobi belo sifundo bafumene ukuba i-injection ye-picamilon yanceda ukubuyisela inani lezilwanyana ze-GABA receptors (iklasi yee-molecule ezithatha i-GABA).
Imeko ephawulwe ngokunyuka komzimba, i-hypokinesia ngamanye amaxesha inxulumene nesifo sika-Parkinson kunye nezinye iingxaki ze-neurological disorders.
Imijelo
Ngenxa yokungabikho kophando, omncinci uyaziwa malunga nokukhuselwa kokusetyenziswa rhoqo kwepiamilon. Nangona kunjalo, kukho inkxalabo yokuba i-picamilon inokubangela inani lemiphumo emibi, njenge -headache , ukubetha, kunye nesisulu. I-Picamilon inokusebenzisana namanye amayeza, njenge-benzodiazepines.
Kubalulekile ukugcina engqondweni ukuba izongezelelo azange zivivinywe ukukhusela kunye nezondlo zokutya zikhululekile. Kwezinye iimeko, loo mveliso inokuhambisa amaxabiso ahluke kwixabiso elichaziweyo kwiyeza ngalinye. Kwezinye iimeko, loo mveliso inokungcoliswa nezinye izinto ezifana nezitye. Kwakhona, ukhuseleko lwezongezelelo kubasetyhini abakhulelweyo, oomama abangabongikazi, abantwana, kunye nalabo abanezifo zonyango okanye abathabatha imishanguzo ayilwanga.
Ezinye iindlela
Ukuba ufuna ukuphucula umsebenzi wengqondo, uninzi lwezonyango zendalo zingasebenzisa enye indawo kwipamiloni. Ngokomzekelo, i-omega-3 fatty acids ifunyenwe ukuphucula umsebenzi wokuqonda, ukugcina imemori, nokukhusela ukuxinezeleka kunye nesifo se-Alzheimer. Ifunyanwe ngokwemvelo kwizinto ezifana neoli ye-flaxse kunye neentlanzi ezinamafutha (kuquka i-salmon, i-sardines, ityhuna, i-mackerel kunye ne-herring), i-omega-3 fatty acids ibuye ithengiswe kwifom yokongeza.
Kukho ubungqina bokuba ezinye iindlela zokwelapha zinganceda ukwandisa amazinga e-GABA ebuchosheni. Ngokomzekelo, uphando oluphambili lubonisa ukuba imifuno efana neva ne- valerian inokuphakamisa amanqanaba e-GABA ngokukhuthaza umdlalo we-GABA okanye ngokunciphisa ukuphazamiseka komzimba we-GABA. Ukongezelela, uphando oluthile lubonisa ukuba ukwenza i-yoga kunokunceda ukwandisa amazinga e-GABA kwaye, kwakhona, ukuphucula isimo sengqondo nokunciphisa uxhalaba.
Kuphi ukuwufumana
Efumaneka ngokubanzi ukuthengwa kwi-intanethi, i-picamilon ithengiswa kwezinye izidakamizwa.
ILizwi
Ngenxa yophando oluncitshisiweyo, kungekudala ukukhuthaza i-picamilon njengonyango nayiphi na imeko.
Kufuneka kuqatshelwe ukuba unyango lwepamilon kunye nokuphepha okanye ukulibazisa ukunakekelwa okuqhelekileyo kunokuba nemiphumo emibi. Ukuba ucinga ngokusetyenziswa kwe-picamilon kwimeko (njengokuba uxinzelelo lwegazi oluphezulu okanye isifo se-Parkinson), qhagamshelana nodokotela wakho ngaphambi kokuba uthathe isilwanyana, njengoko kungenakufaneleka okanye kukhuselekile kubantu abaneemeko ezithile, ezifana nomhlaza.
Imithombo
Kuchmerovskaia TM, Parkhomets PK, Donchenko GV, Obrosova IG, Klimenko AP, Kuchmerovskiĭ NA, Pakirbaeva LV, Efimov AS. "Ukulungiswa kwesifo sikashukela se-neuropathies usebenzisa i-aldose reductase inhibitors kunye ne-pikamilon." Vopr Med Khim. Ngo-1998 uNgo-Dec; 44 (6): 559-64.
I-Akopian VP, i-Balian LS, i-Zakarian NA. "Impembelelo ye-nootropics kwiinguqu ezininzi kwi-corerex ye-cerebral cortex I-GABA (A) i-receptor complexes phantsi kweemeko ze-hypokinesia zokulinga." Eksp Klin Farmakol. 2010 Julayi; 73 (7): 13-5.
Ukuziphendulela: Ulwazi oluqulethwe kule ndawo lujoliswe kwiinjongo zemfundo kuphela kwaye alithathi indawo yeengcebiso, ukuxilongwa okanye unyango ngumgqirha onelayisenisi. Akunakuthetha ukukhusela zonke iindlela zokulondoloza, ukusebenzisana kwezidakamizwa, iimeko kunye nemiphumo emibi. Kufuneka uncede unyango lwangonyango ngokukhawuleza kuyo nayiphi na imiba yempilo uze ubonane nodokotela wakho ngaphambi kokusebenzisa elinye iyeza okanye wenze utshintsho kwi-regimen yakho.