Indlela i-Triptans iyanceda ngayo i-Migraines kunye neyokuyilinda
Ungathatha i-triptan-uyenze uhamba neenxaza kwesikhwama sakho okanye esikhwameni-ukunciphisa ukuhlaselwa kwe-migraine ngokukhawuleza xa ivela. Nangona i-triptan ikhuselekile kwaye ibekezeleke kakuhle, ayilona wonke umntu.
Ukusebenzisa i-Triptan ye-Migraine Relief
I-Triptans isetyenziselwa ukuphatha imodareyitha ezinqamlekileyo, kunye nemigraines emnene engaphenduliyo kwiyeza-counter-counter, ezifana ne-antisteroidal anti-inflammatories .
Zingasetyenziselwa ukuphatha imigraines emnene ukuya kumodareyitha kubantu abangenako ukunyamezela okanye ukuthatha ii-NSAID.
I-Science Behind Triptans
I-Triptans ibopha kwi-serotonin receptors kwingqondo. Ngokusebenzisa i-serotonin receptors, imithwalo yegazi kwingqondo iyancipha kwaye iindlela ezithile zendlela yokuchophaza ingqondo zivaliwe. I-Triptans nayo ikholelwa ukuba isebenza ngokunciphisa amanqanaba e- CGRP -a protein ephakamileyo ngexesha lokuhlaselwa kwe-migraine.
Iindidi ezahlukeneyo
Ii-Triptans zikhangeleka kuba kukho iindlela ezahlukeneyo apho zingathathwa khona. Ngokomzekelo, i-triptan ingathathwa ngomlomo, ngempumlo, okanye ijojowe ngenaliti emathanjeni enomntu omnxeba (obizwa ngokuba yi-injection subcutaneous). Kukho kwakhona i-triptan ebizwa ngokuba yi-Maxalt XLT (rizatriptan) enokutshatyalaliswa ngokukhawuleza emlonyeni womntu kwaye ibandakanyeka nangona umntu ehlanza. Ekugqibeleni, i-Imitrex (i-sumatriptan) inokunikezwa njenge-suppository.
Inguqulelo eninzi yipaki yesikhumba se-triptan.
I-Zecuity (i-sumatriptan) yipatter transmermal esebenzisa ibhetri ehambisa i-sumatriptan ngesikhumba somntu. I-Zekuity, kunye ne-triptans enejojo, ibonakala ngokukodwa kubantu abanentshutshiso kunye nokuhlanza ezinxulumene nemigraines yabo. Oko kuthethwa, ngoJuni ka-2016, i-FDA ithathe uZecuity kwimarike ngenxa yeengxaki zokutshisa okukhulu kunye nezikrakra ezivela kubantu abasebenzisa isixhobo.
Uphando luyaqhubeka.
Iimpembelelo ezingasemva
Ii-Triptans ziyimishanguzo efanelekileyo yokunyanga. Oko kuthethwa, ziyimishanguzo yemithi kwaye kufuneka ukuba ithathwe phantsi kwengqalelo yonyango. Ezinye iziphumo eziqhelekileyo ezichaphazelekayo kunye ne-triptans ziquka:
- I sizathu
- Umtya, intamo, okanye isifuba sesifuba okanye uxinzelelo okanye ukucutha ukuva
- Ukukhawuleza kwentliziyo okanye ukunyuka kwixinzelelo legazi
- Ukukhathala
- Ukuvakalelwa / ukubetha (ikakhulukazi ubuso)
- Ukuvutha kwintsholongwane yolusu
I-Triptans ayinayo yonke into
Kubalulekile ukuhlaziywa kwimbali yakho yezokwelapha kunye nawo onke amayeza akho, kuquka i-add-counter-counter supplements kunye namavithamini, kunye nodokotela wakho. Abanye abantu akufanele bathathe i-triptans kuba bangadala imeko engundoqo yempilo. Ngokomzekelo, akufanele uthathe i-triptan ukuba unembali ye- coronary artery disease , isifo , isifo sesifo se-vascular , ingcinezelo ephezulu yegazi, okanye i- hemiplegic okanye i-basilar migraine.
Ii-Triptans nazo zichasene nabantu abaye bathatha i-monoamine oxidase inhibitors ngokukhawuleza kwaye akufanele kusetyenziswe ngosuku olufanayo njenge-ergotamine okanye i-dihydroergotamine.
Kwakhona, ukudibanisa i-triptan kunye ne-seleotonin reuptake inhibitors (SSRIs) okanye i-norepinephrine reuptake inhibitors (SNRIs) ekhethiweyo ingabangela isifo se-serotonin.
Oku kuyingozi, nangona iimeko ezingavumelekanga ezingabangela iimpawu ezahlukeneyo ezifana:
- kudideka
- ukuxhalaba
- isifo sohudo
- ukuthuka
- ukulahlekelwa kwemali
- ukuthuthumela
- ukuthuthumela
- umkhuhlane
I-Triptans kwi-Women's Childbearing Years
Ngokukhulelwa, i-triptan yicandelo le-C, elithetha ukuba umngcipheko ngokubhekiselele kwinzuzo kufuneka ulinganiswe ngugqirha ngamnye kwisigulane ngasinye. Ngokuxeliswa, ulwazi lwezesayensi ekusebenziseni i-triptans lwe-migraine therapy lucacisiwe-nangona, i-sumatriptan ithathwa njengento ehambelana ne-American Academy of Pediatrics.
Ukuba uthatha i-triptan kunye nesicwangciso sokukhulelwa okanye ukuncelisa, nceda uthetha nodokotela wakho ukuba ufumane isicwangciso sonyango esihle.
ILizwi
Iindaba ezixhasayo malunga ne-triptans kukuba kukho iindlela ezintsha zokuhanjiswa okwangoku, njenge-sumatriptan ulwimi, i-omitriptan inhaler, kunye nomlomo we-rizatriptan ukuchitha ifilimu.
Ii-Triptans zikhetho ezintle zokuphatha imigraines xa inikezelwa phantsi kwengqalelo yonyango. Indlela ekhethekileyo yolawulo iyanceda ngokukhethekileyo ekuphatheni abo bahlanjululwe yi-migraine-nausea ne-vomiting. Yiba ngummeli wempilo yakho ye-migraine kwaye uthethe nogqirha wakho malunga nokuba i-triptan yinto enhle kuwe.
Imithombo:
Ables, A kunye no-Nagubilli R.Ingqungquthela, Ukuxilongwa, kunye noLawulo lweSerotonin Syndrome. I-Phys Physician. 2010 Meyi 1; 81 (9): 1139-1142.
Gilmore B, uMichael M. unyango lwe-Acraine Headache. I-Phys Physician. 2011 Feb 1; 83 (3): 271-280.
IGoldstein J, Smith TR, Pugach N, Griesser J, Sebere T, Pierce M. Iprogram ye-sumatriptan iontophoretic transdermal yonyango olunzulu lwe-migraine. Intloko . 2012 I-Oct; 52 (9): 1402-10.
Hutchinson S, Marmura MJ, Calhoun A, uLucas S, uSilberstein S, Peterlin BL. Ukusetyenziswa kweziNyango zeMigraine eziqhelekileyo kwi-Breast-Feeding Women: Isishwankathelo seNcomelo. Intloko. Ngo-2013 uMatshi; 53 (4): 614-27.
US Food and Drug Administration. (6/2/2016). I-Zecuity (sumatriptan) I-Migraine Patch: Unxibelelwano lokhuseleko lweziyobisi-FDA umngcipheko wokuvavanya nokutshisa.