I-Bone Mineral Density
I-Evista - Yiyiphi into kwaye Yenzani
Ukuba unayo i-osteoporosis okanye i-osteopenia, okanye u-post-menopausal kunye nomngcipheko ophezulu wokuba nomhlaza wesifuba ongenayo, ugqirha wakho unokumisela u-Evista.
I-Evista yigama legama le-raloxifene.
Ekhutshwe ngu-Eli Lilly Corporation, u-Evista ukwandisa ubukhulu bamathambo akho. Yenza umsebenzi wayo ngokulinganisa iziphumo ze-estrogen, i-hormone, phakathi kwezinye izinto, eyakha izicubu zethambo.
Kwaye ngenxa yokukhusela umdlavuza webele, uVevista uyalimaza umphumo we-estrogen kwiisisu zebele - njengokuba i-estrogen kakhulu emzimbeni inokubeka umngcipheko kwesi sifo.
Qaphela ukuba i-Evista yenzelwe abafazi be-postmenopausal , oku kuthetha ukuba ukhulelwe, unesi okanye unako ukukhulelwa, kukulungele ukuthetha nodokotela wakho malunga nokuba le nkunkuma ifanelekile.
I-Evista - Iiklasi zeMithi
I-Evista, (igama eliqhelekileyo: i-raloxifene) yi- SERM , emele ama-modulator-receptor. Iimpawu ze-SERM ziyi-molecule ezidibeneyo eziphazamisa amaziko emathanjeni omzimba wakho (obizwa ngokuthi "i-receptors") ngokuqhelekileyo ayifumana i-estrogen molecules. Ngokuxhomekeka kwimizimba, i-SERM ingakwazi ukuvimba okanye ukuphucula iziphumo ze-estrogen.
Iimpembelelo eziPhakathi
Kodwa i-SERMs, kuquka i-Evista, inokukuchaphazela ngeendlela ezingafunekiyo, ngokunjalo. (Ezi ziya kuba nemiphumo emibi.) Nangona ii-SERM ziyakwazi ukulinganisa i-estrogen ukwenzela ukunceda ukuvelisa ezinye izicubu zethambo, okanye ukuvimbela imiphumo ye-estrogen kwiisisu zebele. , intloko, isisu, intlungu edibeneyo, ukuhlanza kunye / okanye iingxaki zesono.
Kwaye abo bangabamnene. Iziphumo ezibi kakhulu ziyakwenzeka. Ukuba unamava alandelayo, iingcali kwiwebhusayithi ye-Emedicine zibonisa ukuba ufuna unyango ngokukhawuleza:
- Izibonakaliso zempendulo ezithintekayo, umzekelo umlingo, ukuphefumula ubunzima kunye / okanye ukuvuvukala kwemilomo yakho, ubuso, ulwimi okanye umqala.
- Uqala ngokukhawuleza:
- Ubungqina okanye ubuthathaka, ngakumbi kwelinye icala lomzimba
- Intloko, ukudideka, iingxaki nombono wakho, intetho, okanye ukulinganisela
- Intlungu yesifuba, ukukhwehlela, ukuqhuma, ukuphefumula ngokukhawuleza kunye / okanye ukukhawuleza kwenhliziyo
- Ukuvulela ezandleni okanye ezinyaweni
- Izimpawu ezinjenge-Flu: I-Fever, i-chills, isifo somqala kunye nomzimba womzimba
- Ukuphuma kwamagciwane, intlungu yesisu okanye ukunyamezela. Isiqongo esiswini sakho siyabangela ukukhathazeka.
- Ukuvuthwa okubuhlungu, kuquka ukuvutha komlilo
- Intlungu ebuhlungu emva.
Ukusebenzisana kweziyobisi
Ngaphambi kokuba uqale uVevista, kubaluleke kakhulu ukuxelela ugqirha wakho malunga nayiphi na iziyobisi osuke usithatha. Isizathu kukuba ezinye iziyobisi azidibanisi kunye no-Evista, umzekelo u-cholestyramine (amagama e-branded Prevalite kunye neQueestran), okuyiyobisi ye-cholesterol esezantsi.
Abagcini begazi, njenge-Warfarin okanye i-Coumarin bangabonisa ingxaki, ngokunjalo. (Ugqirha wakho unokuyalela uvavanyo oluhlola iprothombrin ukuqinisekisa ukuba iziyobisi ezidibeneyo ziya kukhuseleka kuwe.)
Kwakhona, u-Eli Lilly ucebisa ukuba ungathathi u-Evista ukuba unesifo se-estrogen esithunyelwa ngepilisi, ipaki okanye ngejoyi.
Ezinye iziyobisi ezinokusebenzisana no-Evista ziquka iValium (igama eliqhelekileyo elithi diazepam,) kunye neProglycem (igama eliqhelekileyo elithi diazoxide.) Kunye ne- ibuprofen .
Iimeko ezithile zonyango kunye nemikhwa yokuziphatha ayixubani kakuhle ne-Evista. Okokuqala nangakumbi, ukuba unesifo se-raloxifene, kufuneka uhlale kude no-Evista.
Kuyafana ukuba utshaya, unesifo segazi, unesifo senhliziyo, uxinzelelo lwegazi oluphezulu, isifo sesifo, isifo sesibindi, uye waxabana (nokuba i-TIAs ibala apha), okanye ukuba unesisu nomhlaza ngaphambili.
Qaphela ukuba uluhlu olungasentla lwezilwanyana, iimeko kunye nemikhuba yokuphila ayiphelelanga. Thetha nogqirha wakho ukuze ufumane lonke ulwazi.
> Imithombo:
> RxList. I-Pharmacology Pharmacology - Ukunyuka kwe-12.08.04. Ibuyiswe ngoJulayi 31, 2006.
> RxList. I-Clinical Pharmacology - Indlela yokuSebenza 12.08.04. Ibuyiswe ngoJulayi 31, 2006
> Imithi kunye neDrugs. Emedicine. Kufumaneka: Oktobha 2016. http://www.emedicinehealth.com/drug-raloxifene_oral/article_em.htm
> RxList. Iziphumo eziPhakathi 12.08.04. Ibuyiswe ngoJulayi 31, 2006.
I-Evista, (igama eliqhelekileyo: i-raloxifene) yi- SERM , emele ama-modulator-receptor. Iimpawu ze-SERM ziyi-molecule ezidibeneyo ezibophezela kwi-INTERFERE NEZIMISEBENZI kwii-TISSUES zomzimba (ezibizwa ngokuba yi-receptors) eziqhelekileyo zithola i-estrogen molecules. UKUSEBENZA KWI-TISSUE, I-SERMS IYAVUMA UKUBA KUNYE OKUQHUBILEYO KANYE NOKUBHALISA I-ESTROGEN EFFECT. "Enyanisweni, i-SERM ihlala okanye ishintshele i-estrogen, kwaye ngenxa yoko, inokuguqula umzimba wakho ngendlela echazwe ngasentla. (Ukuchaneka)