Aricept (Donepezil) Amachiza okuPhatha i-Alzheimer's

Yintoni:

Enye yezilwanyana ezisetyenziswa kakhulu ukunyanga iimpawu zesifo se- Alzheimer . I-Aricept i-FDA-ivunyiwe ukuba ibe nemilinganiselo emnene, emodareyithwe , kwaye enzima yesifo.

Ingaba isebenza kanjani:

I-Aricept yi- inhibitor ye-cholineterase evimbela ukuwa kwe- acetylcholine kwingqondo. I-Acetylcholine idlala indima ebalulekileyo kwimemori nokufunda; Amanqanaba aphezulu kwengqondo anceda amangqamuzana omzimba athetha ngokufanelekileyo.

Impumelelo:

Olunye uphando lufumene ukuba i-Aricept inokuyeka ukutshatyalaliswa kweempawu ze-Alzheimer kwiinyanga ezili-6 ukuya kwezi-12 malunga nesiqingatha sabantu abayithathayo. Kwabaninzi, ukuphuculwa kukuncinci, kodwa kulungile. Ubungqina bokuba ngumntu obonisa ukuba i-pesenti encinci yabantu ingazuza ngokugqithiseleyo kule nkunkuma.

Isixa:

I-Aricept ifumaneka kwifomu yeethebhulethi okanye ifom yefomathi ye-tablet ephazamisayo ngomlomo, kwaye iyaqalwa ngo-5 mg ngosuku. Ukuba ukunyamezeleka emva kweeveki ezi-4 ukuya kwezi-6, i-dosage inganyuswa ibe yi-10 mg ngosuku. Unonophelo lwenkonzo yakho yezempilo uya kugqiba umlinganiselo ongcono kuwe okanye wakho othandekayo.

Imiphumela:

Nangona ngokuqhelekileyo ukunyanzeliswa kakuhle, iimpembelelo eziqhelekileyo ziyizicabangela, isifo sohudo, ukunyuka kwamaxesha okunyakaza, ukuhlanza, ukuphazamiseka, ukuphazamiseka kokulala, ukuphazamiseka kwemisipha, ukuphelelwa kwesidlo, ukuphelelwa amandla, ukuphelelwa amandla nokuphelelwa amandla.

Ukubambisana:

Izidakamizwa ezingekho-steroidal ezichasayo (i- NSAID ), ezifana ne-aspirin okanye i-ibuprofen, kufuneka zisetyenziswe ngokuqaphela ngelixa zithatha i-Aricept, ngenxa yengozi yokwanda kwezilonda zesisu .

Ukuqapha:

Qiniseka ukuxelela ugqirha wakho malunga nayiphina imbali okanye iingxaki zangoku zesilonda esiswini , kubandakanywa nawaphi na amayeza athatyathwa ngesimo sesisu. Kwakhona, isichengisi singanciphisa intliziyo yesimo, imeko eyaziwa ngokuba yi- bradycardia .

Umenzi:

I-Aricept yasungulwa ngu-Eisai Inc. kwaye ivunyiwe yi-FDA ngo-1996.

Okwangoku ihanjiswa ngu-Eisai Inc. kwaye ithengiswa nguPfizer Inc.

Generic Iyatholakala:

I-Aricept ifumaneka kwifomu yobudala (HCL).

Imithombo:

Malunga neAricept®. Eisai Inc. kunye nePfizer Inc. 2007. http://www.aricept.com/about/index.aspx

Isifo se-Alzheimer's disease sheet sheet. Izifo ze-Alzheimer's Education and Referral Centre, Isizwe seSizwe sokuguga. NgoJanuwari 15, 2008. http://www.nia.nih.gov/Alzheimers/Publications/medicationsfs.htm

Ionyango ezivunyiweyo ze-FDA ze-Alzheimer's. I-Alzheimer's Association. Julayi 2007. http://www.alz.org/national/documents/topicsheet_treatments.pdf

ScientificWorldJournal. 2013; Ngo-2013: 925702. Ukusebenza kweMemantine, Donepezil, okanye uMbutho wabo kwiZifo eziLungeleleneyo ze-Alzheimer's: Ukuhlaziywa kwezilingo zeCliniki. http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3830825/

-Kuhleliwe ngu-Esther Heerema, MSW