Iinkcukacha NgeRoxin (I-Methocarbamol)

I-Relaxer yeMiscle

I-Robaxin (i-Methocarbamol) iboniswa njengesigxina sokuphumla, unyango lomzimba, kunye nezinye iindlela zokuphucula ukuphazamiseka ezihambelana nezimo ezibuhlungu, ezibuhlungu ezixubileyo. Inkqubo yesenzo se-methocarbamol ayifakwanga ngokucacileyo, kodwa inokuthi ihambelane nezakhiwo zayo zokukhusela. I-Robaxin ayifuni ngokukhawuleza i-muscle muscle kumntu.

Ukungqinelana

I-Robaxin iyaphikiswa kwiigulane ezixhomekeke kwi-methocarbamol okanye nakweyiphi na i-tablet.

Izilumkiso

Ekubeni i-methocarbamol inokuba negalelo eliqhelekileyo le-CNS eliyichukumisayo, izigulane ezitholayo i-Robaxin mazicetyiswe malunga nemiphumo edibeneyo kunye noxinzelelo lwe-CNS.

Ukusetyenziswa okukhuselekileyo kweRobaxin akukasekwa ngokuphathelele kwimiphumo emibi ekuphuculweni komntwana. Kukho iingxelo zentsholongwane kunye nobungqingili obulandelayo emva kokuchaphazeleka kwe-utero kwi-methocarbamol. Ngoko ke, uRobaxin akufanele isetyenziswe kubasetyhini abanakho okanye abakhulelweyo kwaye ngokukodwa ngexesha lokukhulelwa kwangaphambili ngaphandle kokuba isigwebo sogqirha unokuba luncedo ngaphezu kweengozi ezinokwenzeka.

I-Robaxin ingaphazamisa ubuchule bengqondo kunye / okanye emzimbeni efunekayo ekusebenzeni imisebenzi enobungozi, njengemishini yokusebenza okanye ukuqhuba imoto.

Ukuqapha

Izigulane kufuneka zilumkezele ukuba uRoxxin inokubangela ukulala okanye ukutywina, okungathi kunokubangela ukuba bakwazi ukuqhuba izithuthi okanye uomatshini.

Ngenxa yokuba iRoxxin inokuba negalelo eliqhelekileyo le-CNS-ecindezelayo, izigulane kufuneka ziqaphele malunga neziphumo ezidibeneyo ngotywala kunye nabanye abaxinezelekileyo be-CNS.

Izimpembelelo ezimbi

Izimpembelelo ezibi zichazwe ngokuhambelana nokuphathwa kwe-methocarbamol ziquka:

Ukusebenzisana kweDrug kunye neLebhu

I-Robaxin ingavimbela umphumo we-pyridostigmine bromide. Ngoko ke, uRobaxin kufuneka isetyenziswe ngokulumkisa kwizigulane ezine-myasthenia gravis ezifumana ii-anticholinesterase agents.

I-Methocarbamol ingabangela ukuphazamiseka kombala kwiimvavanyo ezithile zokuhlola i-5-hydroxyindoleacetic acid.

I-Carcinogenesis, i-Mutagenesis, Ukungonakali kobutyebi

Izifundo zexesha elide ukuvavanya i-carbagenic ye-Robaxin ayinakwenziwa. Akukho zifundo ezenziweyo ukuvavanya umphumo weRobaxin kwi-mutagenesis okanye amandla ayo okuphazamisa ukuzala.

Ukukhulelwa

Izifundo zokuzaliswa kwezilwanyana azizange zenziwe nge-methocarbamol.

Akukwazanga nokuba ingaba i-methocarbamol ingabangela ingozi yomntwana xa ilawulwa kumfazi okhulelweyo okanye inokuchaphazela amandla okuvelisa. I-Robaxin kufuneka inikwe umfazi okhulelweyo kuphela xa kufuneka ngokucacileyo.

Ukusetyenziswa okukhuselekileyo kweRobaxin akukasekwa ngokuphathelele kwimiphumo emibi ekuphuculweni komntwana. Kukho iingxelo zentsholongwane kunye nobungqingili obulandelayo emva kokuchaphazeleka kwe-utero kwi-methocarbamol. Ngoko ke, uRobaxin akufanele isetyenziswe kubasetyhini abanakho okanye abakhulelweyo kwaye ngokukodwa ngexesha lokukhulelwa kwangaphambili ngaphandle kokuba isigwebo sogqirha unokuba luncedo ngaphezu kweengozi ezinokwenzeka.

Oomama abanesihlengikazi

I-Methocarbamol kunye / okanye i-metabolites yayo ixutywe kubisi lwezinja; Nangona kunjalo, awaziwa ukuba i-methocarbamol okanye i-metabolites yayo ixutywe ebisi lomntu. Ngenxa yokuba ezininzi izidakamizwa zixutywa ngobisi, kufuneka uqaphele xa uRoxxin ilawulwa ngumfazi onesihlengikazi.

Ukusetyenziswa kwezilwanyana

Ukhuseleko kunye nokusebenza kwe-Robaxin kwizigulana zezilwanyana ezingaphantsi kweminyaka eyi-16 azizange zenziwe.

Ngaphezulu

Ulwazi oluthile lufumaneka kwi-toxicity ye-methocarbamol. Ukugqithiswa kwe-methocarbamol ngokuqhelekileyo kudibaniswa notywala okanye ezinye izidumbu zakwa-CNS kwaye ziquka ezi zilandelayo:

Kwimeko yamava okuthengisa, ukufa kwabikwa ngokugqithisileyo kwe-methocarbamol yedwa okanye phambi kwezinye iincinci ze-CNS, iziyobisi okanye iziyobisi zengqondo. Ulawulo lokugqithisa ngokwexesha kubandakanywa unyango olungumqondiso kunye nokuxhasa.

Gcina i-Robaxin kwiqondo lokushisa lokulala, phakathi kwe-20 ° C no-25 ° C (68 ° F no-77 ° F).

Umthombo:

I-US yokuLawula kunye nokuLawula iDrug, i-NDA 11-011 / S-070/071