I-Methimazole, i-Carbimazole kunye nePropylthiouracil / i-PTU
Xa isifo se-thyroid siba namandla - imeko eyaziwa ngokuba yi-hyperthyroidism - i-gland ikhiqiza i-hormone ephezulu ye-thyroid. Oku, kunokubangela iimpawu ezahlukahlukeneyo, kubandakanywa ukuqhuma okukhawulezayo, uxinzelelo lwegazi oluphezulu, ukuxhalaba, ukulala, ukuthuthumela, ukulahleka kwesisindo, ukuhanjiswa, kunye nemininzi yempawu ye-metabolism engaphaya, kunye neengqungquthela ezingapheliyo kunye namalungu.
Unyango oluphambili lwe-hyperthyroidism ludidi lweemithi zonyango ezibizwa ngokuba yiziyobisi ze-antithyroid. Iziyobisi ze-Antithyroid nazo zibizwa ngokuba yi-thioamide. Ziyizidakamizwa ezisetyenziselwa ukhathaza i-thyroid engasebenzi - hyperthyroidism - kubandakanywa xa i-thyroid ingasebenzi ngaphezu kweSifo se-Graves, i-goiter ye-multinodular goiter, okanye ii-nodules ezinobuthi.
Izidakamizwa ze-Antithyroid zisebenza ngokuthintela i-thyroid gland ukukwazi ukuvelisa ezimbini ezibalulekileyo ze-thyroid i-thyroxine (T4) kunye ne-triiodothyronine (T3).
Izidakamizwa eziphambili ze- antithyroid e-United States zifumaneke nge-methimazole kunye nepropylthiouracil (PTU). Ngaphandle kwe-United States, ukhetho luyimethimazole, carbimazole, kunye ne-PTU.
Methimazole
I-antithyroid yezidakamizwa i-methimazole inhibitshi ye-thyroid ekusebenziseni i-iodine-ngokuqhelekileyo ukusuka ekudleni okanye kwi-supplements-ukuvelisa i-hormone ye-thyroid. Ingumuthi ngokuqhelekileyo uthathwa kanye ngosuku ngemigulane.
Ngamanye amaxesha i-Methimazole ibizwa ngokuba yi-thiamazole.
Eli seziyobisi lisetyenziswe kwihlabathi jikelele kwaye isilwanyana esiphambili se-antithyroid esisetyenzisiweyo e-United States, apho sitholakala ngaphantsi kwegama leTapazole.
Abakhiqizi abaningana banikezela uhlobo oluthile lwe-methimazole.
ICarbimazole
I-Carbimazole yilezi zizaziso, xa zilawulwe, ziguqulwa kwi-drug methimazole emzimbeni, kwaye ngoko ke zifana nezenzo.
I-brand eyaziwayo kakhulu ye-carbimazole yi-Neomercazole.
I-Neomercazole libizwa ngegama lomthi we-carbimazole kwaye lenziwe yi-Amdipharm International (UK). Esi sigqirha sagunyaziwe ngo-2004, kwaye sithengiswa e-UK naseYurophu, kodwa ayifumaneki okanye imiselwe eMelika. Uyakwazi ukubona i datasheet kwi- Neomercazole apha. Nazi ezinye iinkcukacha ezongezelelweyo malunga neNomercazole.
- Iwebhusayithi kaMenzi weziyobisi: i-Amdipharm
- Ulwaziso loLwazi
Neomercazole Izithako : i-carbimazole Ph.Eur; lactose; isitashi sombona; sucrose; i-magnesium stearate; sucrose; talc; i-gum acacia; i-ferric oxide; propyl hydroxybenzoate; ne gelatin.
Amandla afumanekayo : 5 mg
Amanye amaBrama / amagama: I- Carbimazole ifumaneka kwamanye amazwe aseYurophu nase-Asia phantsi kwamagama alandelayo alandelayo: Atirozidina, Basolest, CG1, i-Carbimazole Spofa, iCarbotiroid, i-Mertiran, i-Neo-Mercazole, i-Neo-Thyreostat, i-Neo-Tireol neTyrazol.
Propylthiouracil / PTU
Indlela i-PTU yenza ukuba i -roid ye-hormone ye-thyroid igqithise kakhulu i-thyroid i-hormone ye-thyroid. Kwakhona kuvimbela ukuguqulwa kwe-hormone ye-thyroid iT4 kwi-T3. I-PTU inexesha elifutshane elibambeleyo, ngoko ke izigulane ezithatha le mayeza ziyalwa ukuba zithathe iyeza zimbini ukuya kathathu ngosuku ukuya kumazinga e-hormone ye-thyroid.
I-PTU ineempembelelo ezingaphezulu kunezinye iziyobisi ezixutyushwa apha, kwaye yiyobisi ekhethiweyo ye-hyperthyroidism kuphela kwiimeko ezimbalwa (ngexesha lokukhulelwa kwangaphambili, isifo esiqatha se-thyroid kwaye xa isigulane sibhekene nemiphumo emibi ephuma kwi-methimazole).
EUnited States, kuphela i-PTU yendalo ekhoyo; akukho namagama e-brand ye-PTU athengiswayo e-United States. Inani labakhiqizi livelisa i-PTU.
Iinkcukacha ezithe xaxe
Funda kabanzi malunga ne-hyperthyroidism kunye nonyango lwawo, kubandakanywa iziyobisi zakwa-antithyroid, kwezi zixhobo:
- Hyperthyroidism | Izifo zeMangcwaba | I-Thyroid engasebenzi
- Izifo zeMangcwaba kunye ne-Hyperthyroidism 101
- I-Hyperthyroidism Iingozi / Iimpawu zokuHlola
- Ingozi yeeNgcwaba kunye neHyperthyroidism
- Imibuzo Ebuzwa Ngokuphindaphindiweyo kwi-Hyperthyroidism ne-Graves 'Diesase
- Iindlela ezintathu zokuphatha i-Hyperthyroidism
Imithombo:
I-Med Med, iDaily Food and Drug Administration, i-Online Med
I-FDA Inxibelelwano loKhuseleko lweMithi: I-Box Boxed entsha kwi-injection enkulu yesibindi kunye nepropylthiouracil, uEpreli 21, 2010, i-Intanethi
Ross, Douglas MD, "Ulwazi olunomonde: Izidakamizwa ze-Antithyroid," UpToDate . Kuhlaziywa ngokutsha: ngoNovemba 13, 2009